Friday, January 25, 2013

Loratadine


KP Wellness

13:57  -  Public
Loratadine is a second-generation H1 histamine antagonist drug used to treat allergies.  marketed for its non-sedating properties. In a version named Claritin-D or Clarinase, it is combined with pseudoephedrine, a decongestant; this makes it useful for colds as well as allergies but adds potential side-effects of insomnia, anxiety, and nervousness.

Loratadine is indicated for the symptomatic relief of allergy such as hay fever (allergic rhinitis), urticaria (hives), and other skin allergies. For allergic rhinitis (hay fever), loratadine is effective for both nasal and eye symptoms: sneezing, runny nose, itchy or burning eyes.

In the U.S., it is classified as category B in pregnancy, meaning that animal reproduction studies have failed to demonstrate a risk to the fetus, and there are no adequate and well-controlled studies in pregnant women.

while taking loratadine should avoid the use of alcohol as it can cause excessive drowsiness.

Loratadine's peak effect occurs in 1–2 hours, and its biological half-life is on average 8 hours (range 3–20 hours)

Substances that act as inhibitors of the CYP3A4 enzyme such as ketoconazole, erythromycin, cimetidine and furanocoumarin derivates (found in grapefruit) lead to increased plasma levels of loratadine.  
Padma Dorje originally shared this post:
It helped me a lot today.
Loratadine - Wikipedia, the free encyclopedia »
Systematic (IUPAC) name. Ethyl 4-(8-chloro-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-ylidene)-1-piperidinecarboxylate. Clinical data. Trade names, Claritin. AHFS/Drugs.com, monograph. Medl...
 

KP Wellness

13:50  -  Public
Chau Le - Joy Le originally shared this post:
#Allergic  #rhinitis  is  very  common. Seasonal #allergicRhinitis is most commonly caused by pollens and spores. Flowering shrub and tree pollens are most common in the spring, flowering plants and grasses in the summer, and ragweed and molds in the fall. Dust, house-hold mites, air pollution, and pet dander may produce year-round symptoms, termed “perennial rhinitis.”
Allergic  rhinitis  is  caused  by  exposure  to  an  airborne allergen  in  a  predisposed  individual.  Activation  of  both humoral (B-cell) and cytotoxic (T-cell) immune responses with  subsequent  allergen-specific  IgE  responses  causes release  of  inflammatory  mediators.  The  response  is
increased as antigen is passed to regional lymph nodes for greater  T-cell  activation.  Interleukin  and  cytokine  release causes specific activation of mast cells, eosinophils, plasma cells, basophils and other T-cells. Many of these circulating cells  then  migrate  into  the  nasal  and  ocular  epithelium
where  they  contribute  directly  to  symptoms  through proinflammatory  mediators,  including  histamine,  prosta-glandins, and kinins.

          Clinical Findings
The  symptoms  of “hay  fever”  are  similar  to  those  of  viral rhinitis  but  are  usually  persistent  and  may  show  seasonal variation.  Nasal  symptoms  are  often  accompanied  by  eye irritation,  pruritus,  conjunctival  erythema,  and  excessive tearing. Many patients will note a strong family history of atopy or allergy.
The  clinician  should  be  careful  to  distinguish  allergic rhinitis from nonallergic or vasomotor rhinitis. Vasomotor rhinitis  is  caused  by  increased  sensitivity  of  the  vidian nerve  and  is  a  common  cause  of  clear  rhinorrhea  in  the elderly. Often patients will report that they have troubling rhinorrhea in response to numerous nasal stimuli, includ-ing warm or cold air, odors or scents, light, or particulate matter. On physical examination, the mucosa of the turbinates is  usually  pale  or  violaceous  because  of  venous  engorge-ment. This is in contrast to the erythema of viral rhinitis. Nasal polyps, which are yellowish boggy masses of hyper-trophic mucosa, are associated with long-standing allergic rhinitis.

Treatment

A. Intranasal Corticosteroids
Intranasal  corticosteroid  sprays  have  revolutionized  the treatment  of  allergic  rhinitis.  Evidence-based  literature reviews show that these are more effective—and frequently less expensive—than nonsedating antihistamines. Patients should be reminded that there may be a delay in onset of relief  of  2  or  more  weeks.  Corticosteroid  sprays  may  also
shrink hypertrophic nasal mucosa and nasal polyps, thereby providing an improved nasal airway and osteomeatal com-plex  drainage.  Because  of  this  effect,  intranasal  corticos-teroids are critical in treating allergy in patients prone to recurrent  acute  bacterial  rhinosinusitis  or  chronic  rhi-nosinusitis.  There  are  many  available  preparations, including  beclomethasone  (42  mcg/spray  twice  daily  per nostril),  flunisolide  (25  mcg/spray  twice  daily  per  nos-tril),  mometasone  furoate  (200  mcg  once  daily  per  nos-tril),  budesonide  (100  mcg  twice  daily  per  nostril)  and fluticasone propionate (200 mcg once daily per nostril). All intranasal corticosteroids are considered equally effective. Probably the most critical factor is compliance with regu-lar  use  and  proper  introduction  into  the  nasal  cavity.  In order  to  deliver  medication  to  the  region  of  the  middle
meatus,  proper  application  involves  holding  the  bottle straight up with the head tilted forward and pointing the bottle toward the ipsilateral ear when spraying. Side effects are  limited  and  the  most  annoying  is  epistaxis.  Some experts  believe  that  this  is  related  to  incorrect  delivery  of the drug to the nasal septum.

B. Antihistamines
Treatment of allergic and perennial rhinitis has improved in recent years. Antihistamines offer temporary, but imme-diate, control of many of the most troubling symptoms of allergic  rhinitis.  Over-the-counter  antihistamines  include nonsedating  #loratadine  (10  mg  orally  once  daily)  and minimally  sedating  cetirizine  (10  mg  orally  once  daily). Brompheniramine  or  chlorpheniramine  (4  mg  orallyevery 6–8 hours, or 8–12 mg orally every 8–12 hours as asustained-release  tablet)  and  clemastine  (1.34–2.68  mg
orally twice daily) may be less expensive, although usually associated  with  some  drowsiness.  Prescription  oral H1-receptor  antagonists  include  fexofenadine  (60  mgtwice daily or 120 mg once daily) and desloratadine (5 mg  once  daily).  Fexofenadine  appears  to  be  nonsedating;
desloratadine  is  minimally  sedating.  Also  shown  to  be effective  in  randomized  trials  are  ebastine  (10–20  mg orally  once  daily)  and  misolastine  (10  mg  orally  once daily).  The  H1-receptor  antagonist  antihistamine  nasal spray azelastine (1–2 sprays per nostril daily) has also been shown to be effective in a randomized trial. Topical #nasal
sprays  are  particularly  useful  in  patients  who  experience
side effects, mostly xerostomia and sedation, of oral anti-histamines. Many patients who find initial benefit from an antihistamine complain that allergy symptoms eventually return after several months of use. In such patients, typi-cally with perennial allergy problems, antihistamine toler-ance  seems  to  develop  and  alternating  effective antihistamines  periodically  can  control  symptoms  over the long term.

C. Adjunctive Treatment Measures
In  addition  to  intranasal  corticosteroid  sprays  and  anti-histamines, including H1-receptor antagonists, the litera-ture supports the use of antileukotriene medications such as  montelukast  (10  mg/d  orally)  alone  or  with  #cetirizine (10 mg/d orally) or loratadine (10 mg/d orally). There are
proinflammatory effects of cysteinyl leukotrienes in upper airway disease, including allergic rhinitis, and hyperplas-tic  polyposis,  and  sinusitis.  Improved  nasal  rhinorrhea, sneezing, and congestion are seen with the use of leukot-riene  receptor  antagonists,  often  in  conjunction  with
antihistamines. Cromolyn sodium and sodium nedocro-mil  are  also  useful  adjunct  agents  for  allergic  rhinitis.
They work by stabilizing mast cells and preventing proin-flammatory  mediator  release.  They  are  not  absorbed  by the  gastrointestinal  tract  but  do  function  topically  and have  very  few  side  effects.  The  most  useful  form  of  cro-molyn  is  probably  the  ophthalmologic  preparation;  the nasal preparation is not nearly as effective as inhaled cor-ticosteroids.  Intranasal  cromolyn  is  cleared  rapidly  and must  be  administered  four  times  daily  for  continued relief of symptoms.

Intranasal anticholinergic agents, such as ipratropium bromide  0.03%  or  0.06%  sprays  (42–84  mcg  per  nostril three times daily), may be helpful adjuncts when rhinor-rhea  is  a  major  symptom.  Ipratropium  nasal  sprays  are not  as  effective  as  intranasal  corticosteroids  for  treating
allergic  rhinitis  but  are  useful  for  treating  vasomotor rhinitis. Avoiding or reducing exposure to airborne allergens is the most effective means of alleviating symptoms of aller-gic rhinitis. Depending on the allergen, this can be extremely difficult.  Maintaining  an  allergen-free  environment  by
covering pillows and mattresses with plastic covers, substi-tuting  synthetic  materials  (foam  mattress,  acrylics)  for animal  products  (wool,  horsehair),  and  removing  dust-collecting household fixtures (carpets, drapes, bedspreads,wicker)  is  worth  the  attempt  to  help  more  troubled
patients. Air purifiers and dust filters may also aid in main-taining  an  allergen-free  environment.  Nasal  saline  irriga-tions  are  a  useful  adjunct  in  the  treatment  of  allergic rhinitis to mechanically flush the allergens from the nasal cavity. Though debated, there is no clear benefit to hyper-tonic  saline  over  commercially  available  normal  saline preparations  (eg,  Ayr  or  Ocean  Spray).  When  symptoms are extremely bothersome, a search for offending allergens may prove helpful. This can either be done by serum radio-allergosorbent  test  (RAST)  testing  or  skin  testing  by  an
allergist.In  some  cases,  allergic  rhinitis  symptoms  are  inade-quately  relieved  by  medication  and  avoidance  measures. Often, such patients have a strong family history of atopy and  may  also  have  lower  respiratory  manifestations  such as  allergic  #asthma.  Referral  to  an  allergist  may  be  appro-priate  for  consideration  of  immunotherapy.  This  treat-ment  course  is  quite  involved,  with  proper  identification of  offending  allergens,  progressively  increasing  doses  of allergen(s) and eventual maintenance dose administration over  a  period  of  3–5  years.  Immunotherapy  has  been proven  to  reduce  circulating  IgE  levels  in  patients  with allergic  rhinitis  and  reduce  the  need  for  allergy  medica-tions. While oral allergen exposure is actively being inves-tigated,  currently  the  primary  mode  of  allergen  exposure is  by  subcutaneous  injection.  Treatments  are  given  at  a suitable medical facility with monitoring following treat-ment because of the risk of anaphylaxis during dose esca-lation.  Local  reactions  are  common  and  usually self-limited. 
 

KP Wellness

13:34  -  Public
Perla Cavazos originally shared this post:
The Word for Today: Loratadine. Pronunciation: /lə-ˈrat-ə-ˌdēn, -ˌdīn/ It is used to temporarily relieve the symptoms of hay fever (allergy to pollen, dust, or other substances in the air) and other allergies. These symptoms include sneezing, runny nose, and itchy eyes, nose, or throat.
 

KP Wellness

13:34  -  Public
Bernard Doove originally shared this post:
Hayfever was making me miserable - sneezing constantly, runny nose, constant itching, and by Wednesday I was gasping for breath. Got some Loratadine from the pharmacy on Thursday and it's like a miracle cure.  Best I've felt in weeks, and nary a sniffle.  It's nice to find a medicine that actually works as advertised.
 

KP Wellness

13:33  -  Public
ChristianVision Eye Services to Haiti originally shared this post:
Clinic Wed-34pp |Featured|: Had a visit from 4C pharm reps today. They left a spread. Not sure how much I'll use.

Pictured
Ophthalnol  Artificial Tear
Ophthalmid  10% Sulfacetamide
Myoxan  Chlorzoxazone/Acetaminophen
Lora  Loratadine
Lora Sinus  Loratadine/Psuedoephedrine
Doralil  Naproxen/Acetaminophen
 

KP Wellness

13:32  -  Public
You should not drink alcohol while on the med as it will cause you to feel even more sleepy and drowsy.
 If you do not have the telltale signs of seasonal allergy, don’t take Loratadine.

Loratadine side effects can include symptoms of allergy, like watery eyes, dripping sinuses, itching and sneezing. If you have these side effects, you may or may not be allergic to the medication itself.

If your heart begins to beat faster, even while you are in a resting position, you may not be able to continue the course of treatment. If your skin becomes unhealthy looking, or takes on a yellowish tone, this is another possible side effect.
rama chandra originally shared this post:
LORATADINE SIDE EFFECTS – CAN THEY BE AVOIDED?
 
LORATADINE SIDE EFFECTS – CAN THEY BE AVOIDED? ~ HEALTH TIPS »
Loratadine side effects almost always disappear within a few days of being on this drug. Loratadine and Claritin are technically the same drugs, but the first one is only available by prescription. Th...
 

KP Wellness

13:28  -  Public
RESPIRATORY

Dimetapp
chlorpheniramine
clemastine
diphenhydramine
pseudoephedrine
phenylephrine
loratadine
Your Health originally shared this post:
OTC Drugs List  



KP Wellness

14:22  -  Public
Children’s Claritin Chewables promise to provide 24 hours of allergy relief without drowsiness.
In My Bag originally shared this post:
In My Bag » Upcoming review: Children’s Claritin Chewables »
Ugh, allergies. I'm suffering pretty badly this year, and it's only the end of March, so for all intents and purposes spring has barely begun (though spring
 

KP Wellness

14:08  -  Public
You know what to do between Seasonal allergies and flu.
Erin Coyne originally shared this post:
Dear Claritin:

I know you're working because I can breathe again, and because my eye finally stopped watering.....

But what's with the runny nose and all the sneezing?!

Get it together.

Love,
Erin
 

KP Wellness

14:05  -  Public
Abrazo Health Care originally shared this post:
Watch your kids for allergy symptoms

You know the common symptoms of allergies: red eyes, sinus pressure, headache, scratchy throat, sneezing. But not all allergies kids face are that obvious. Be on the lookout for clues such as unexplained rashes or cold symptoms that last for more than a week.

Most allergy symptoms in the respiratory tract respond well to over-the-counter (OTC) medicines, like Claritin, Zyrtec. For skin conditions, try hydrocortozone creams. If symptoms continue, you may want to make an appointment with your pediatrician.
Image credit: Characteristicly Noah by Sherif Salama http://www.flickr.com/photos/mazboot/286226908/
 

KP Wellness

14:03  -  Public
Seasonal allergies almost always cause people to feel congested, stuffy and produce excess mucus. Additionally, you may have watery eyes, redness and irritation around the nasal passages and develop a slight fever. By contrast, flu suffers have body aches, extremely high body temperatures and severe sore throats.

Note that natural allergy remedies will not work on flu or common cold sufferers.

http://healthwalaa.blogspot.com/2012/12/seasonal-allergy-symptoms-vs-common.html
SEASONAL ALLERGY SYMPTOMS VS COMMON COLD AND FLU ~ HEALTH TIPS »
If you have recently been experiencing sneezing and runny nose, these might as well be seasonal allergy symptoms. However, you may also have either a cold or the flu. Knowing the difference between th...






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